Agency
National Institute of Health (NIH)
Institute
National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK)
Type
Research Project (R01)
Project #
3R01DK015410-16S2
Application #
3225390
Study Section
(SRC)
Project Start
1974-09-01
Project End
1988-03-31
Budget Start
1987-09-01
Budget End
1988-03-31
Support Year
16
Fiscal Year
1987
Total Cost
Indirect Cost
Name
University of California San Diego
Department
Type
Schools of Arts and Sciences
DUNS #
077758407
City
La Jolla
State
CA
Country
United States
Zip Code
92093
Moore, Sandra Blaj; van der Hoek, Joost; de Capua, Antonia et al. (2005) Discovery of iodinated somatostatin analogues selective for hsst2 and hsst5 with excellent inhibition of growth hormone and prolactin release from rat pituitary cells. J Med Chem 48:6643-52
Moore, S B; Grant, M; Rew, Y et al. (2005) Synthesis and biologic activity of conformationally constrained analogs of L-363,301. J Pept Res 66:404-22
Kelleman, Audrey; Mattern, Ralph-Heiko; Pierschbacher, Michael D et al. (2003) Incorporation of thioether building blocks into an alphavbeta3-specific RGD peptide: synthesis and biological activity. Biopolymers 71:686-95
Del Valle, Juan R; Goodman, Murray (2003) Asymmetric hydrogenations for the synthesis of Boc-protected 4-alkylprolinols and prolines. J Org Chem 68:3923-31
Jiang, S; Gazal, S; Gelerman, G et al. (2001) A bioactive somatostatin analog without a type II' beta-turn: synthesis and conformational analysis in solution. J Pept Sci 7:521-8
Falb, E; Salitra, Y; Yechezkel, T et al. (2001) A bicyclic and hsst2 selective somatostatin analogue: design, synthesis, conformational analysis and binding. Bioorg Med Chem 9:3255-64
Goodman, M; Zapf, C; Rew, Y (2001) New reagents, reactions, and peptidomimetics for drug design. Biopolymers 60:229-45
Li, H; Jiang, X; Goodman, M (2001) Synthesis, conformational analysis and biological activities of lanthionine analogs of a cell adhesion modulator. J Pept Sci 7:82-91
Rueter, J K; Mattern, R H; Zhang, L et al. (2000) Syntheses and biological activities of sandostatin analogs containing stereochemical changes in positions 6 or 8. Biopolymers 53:497-505
Li, H; Jiang, X; Howell, S B et al. (2000) Synthesis, conformational analysis and bioactivity of Lan-7, a lanthionine analog of TT-232. J Pept Sci 6:26-35

Showing the most recent 10 out of 40 publications