Funding Agency

Agency
National Institute of Health (NIH)
Institute
National Institute on Drug Abuse (NIDA)
Type
Method to Extend Research in Time (MERIT) Award (R37)
Project #
5R37DA012394-06
Application #
6788694
Study Section
Special Emphasis Panel (NSS)
Program Officer
Rapaka, Rao
Project Start
1999-05-15
Project End
2007-04-30
Budget Start
2004-05-01
Budget End
2005-04-30
Support Year
6
Fiscal Year
2004
Total Cost
$255,139
Indirect Cost

  Institution

Name
University of Arizona
Department
Pharmacology
Type
Schools of Medicine
DUNS #
806345617
City
Tucson
State
AZ
Country
United States
Zip Code
85721

  Publications

Petrov, Ravil R; Lee, Yeon Sun; Vardanyan, Ruben S et al. (2013) Effect of anchoring 4-anilidopiperidines to opioid peptides. Bioorg Med Chem Lett 23:3434-7
Lee, Yeon Sun; Fernandes, Steve; Kulkarani, Vinod et al. (2010) Design and synthesis of trivalent ligands targeting opioid, cholecystokinin, and melanocortin receptors for the treatment of pain. Bioorg Med Chem Lett 20:4080-4
Lee, YeonSun; Petrov, Ravil; Kulkarni, Vinod et al. (2009) Development of mu/delta opioid ligands: enkephalin analogues containing 4-anilidopiperidine moiety. Adv Exp Med Biol 611:517-8
Agnes, Richard S; Ying, Jinfa; Kover, Katalin E et al. (2008) Structure-activity relationships of bifunctional cyclic disulfide peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors. Peptides 29:1413-23
Lee, Yeon Sun; Agnes, Richard S; Cain, James P et al. (2008) Opioid and melanocortin receptors: do they have overlapping pharmacophores? Biopolymers 90:433-8
Shinoda, Katsumi; Hruby, Victor J; Porreca, Frank (2007) Antihyperalgesic effects of loperamide in a model of rat neuropathic pain are mediated by peripheral delta-opioid receptors. Neurosci Lett 411:143-6
Lee, Yeon Sun; Petrov, Ravil; Park, Chad K et al. (2007) Development of novel enkephalin analogues that have enhanced opioid activities at both mu and delta opioid receptors. J Med Chem 50:5528-32
Lee, Yeon Sun; Nyberg, Joel; Moye, Sharif et al. (2007) Understanding the structural requirements of 4-anilidopiperidine analogues for biological activities at mu and delta opioid receptors. Bioorg Med Chem Lett 17:2161-5
Lee, Yeon Sun; Agnes, Richard S; Davis, Peg et al. (2007) Partial retro-inverso, retro, and inverso modifications of hydrazide linked bifunctional peptides for opioid and cholecystokinin (CCK) receptors. J Med Chem 50:165-8
Agnes, Richard S; Lee, Yeon Sun; Davis, Peg et al. (2006) Structure-activity relationships of bifunctional peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors. J Med Chem 49:2868-75

Showing the most recent 10 out of 17 publications