Agency
National Institute of Health (NIH)
Institute
National Institute on Drug Abuse (NIDA)
Type
Research Project (R01)
Project #
1R01DA004087-01A1
Application #
3209149
Study Section
(DABB)
Project Start
1987-01-01
Project End
1989-12-31
Budget Start
1987-01-01
Budget End
1987-12-31
Support Year
1
Fiscal Year
1987
Total Cost
Indirect Cost
Name
University of Michigan Ann Arbor
Department
Type
Schools of Medicine
DUNS #
791277940
City
Ann Arbor
State
MI
Country
United States
Zip Code
48109
Hillhouse, Todd M; Porter, Joseph H (2015) A brief history of the development of antidepressant drugs: from monoamines to glutamate. Exp Clin Psychopharmacol 23:1-21
Bender, Aaron M; Clark, Mary J; Agius, Michael P et al. (2014) Synthesis and evaluation of 4-substituted piperidines and piperazines as balanced affinity ? opioid receptor (MOR) agonist/? opioid receptor (DOR) antagonist ligands. Bioorg Med Chem Lett 24:548-51
Mosberg, Henry I; Yeomans, Larisa; Harland, Aubrie A et al. (2013) Opioid peptidomimetics: leads for the design of bioavailable mixed efficacy ýý opioid receptor (MOR) agonist/ýý opioid receptor (DOR) antagonist ligands. J Med Chem 56:2139-49
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Purington, Lauren C; Sobczyk-Kojiro, Katarzyna; Pogozheva, Irina D et al. (2011) Development and in vitro characterization of a novel bifunctional ?-agonist/?-antagonist opioid tetrapeptide. ACS Chem Biol 6:1375-81
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