|
Brandt, M E; Puett, D; Garola, R et al. (1988) Aromatase and aromatase inhibitors: from enzymology to selective chemotherapy. Prog Clin Biol Res 262:65-84
|
|
Heston, W D; Yang, C R; Pliner, L et al. (1987) Cytotoxic activity of a polyamine analogue, monoaziridinylputrescine, against the PC-3 human prostatic carcinoma cell line. Cancer Res 47:3627-31
|
|
Heston, W D; Watanabe, K A; Pankiewicz, K W et al. (1987) Cytotoxic and non-cytotoxic N-alkyl derivatives of putrescine: effect on polyamine uptake and growth of prostatic cancer cells in vitro. Biochem Pharmacol 36:1849-52
|
|
Naritoku, D K; Levine, J A; Covey, D F et al. (1987) Effects of anticonvulsant and convulsant gamma-butyrolactones and thiobutyrolactones on GABA-mediated chloride uptake. Biochem Pharmacol 36:797-800
|
|
Covey, D F; McMullan, P C; Weaver, A J et al. (1986) Inactivation of Streptomyces hydrogenans 20 beta-hydroxysteroid dehydrogenase by an enzyme-generated ethoxyacetylenic ketone in the presence of a thiol. Biochemistry 25:7288-94
|
|
Auchus, R J; Covey, D F (1986) Mechanism-based inactivation of 17 beta,20 alpha-hydroxysteroid dehydrogenase by an acetylenic secoestradiol. Biochemistry 25:7295-300
|
|
Beusen, D D; Kalman, B L; Covery, D F (1986) Role of substrate conformational features in the stereospecificity of aromatase. Biochemistry 25:662-7
|
|
Covey, D F; Hood, W F; McMullan, P C (1986) Studies of the inactivation of human placental aromatase by 17 alpha-ethynyl-substituted 10 beta-hydroperoxy and related 19-nor steroids. Biochem Pharmacol 35:1671-4
|
|
Levine, J A; Ferrendelli, J A; Covey, D F (1986) Alkyl-substituted thiolo-, thiono-, and dithio-gamma-butyrolactones: new classes of convulsant and anticonvulsant agents. J Med Chem 29:1996-9
|
|
Heston, W D; Uy, L; Fair, W R et al. (1985) Cytotoxic activity of aziridinyl putrescine enhanced by polyamine depletion with alpha-difluoromethylornithine. Biochem Pharmacol 34:2409-10
|
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