Active-Side-Directed Inhibitors of Gar Transformylase

Caperelli, Carol A.

Abstract

Funding Agency

• Agency: National Institute of Health (NIH)
• Institute: National Cancer Institute (NCI)
• Type: Research Project (R01)
• Project #: 5R01CA028312-05
• Application #: 3168067
• Study Section: Bio-Organic and Natural Products Chemistry Study Section (BNP)
• Project Start: 1980-02-01
• Project End: 1985-12-31
• Budget Start: 1985-07-01
• Budget End: 1985-12-31
• Support Year: 5
• Fiscal Year: 1985

Institution

• Name: New York University
• Type: Schools of Arts and Sciences
• DUNS #: 004514360
• City: New York
• State: NY
• Country: United States
• Zip Code: 10012

Publications

Caperelli, C A; Price, M F (1988) Carbocyclic glycinamide ribonucleotide is a substrate for glycinamide ribonucleotide transformylase. Arch Biochem Biophys 264:340-2

Caperelli, C A; Conigliaro, J (1986) Synthesis of 10-acetyl-5,8-dideazafolic acid: a potent inhibitor of glycinamide ribonucleotide transformylase. J Med Chem 29:2117-9

Caperelli, C A (1985) Mammalian glycinamide ribonucleotide transformylase: purification and some properties. Biochemistry 24:1316-20

Lloyd, R D; Jones, C W; Mays, C W et al. (1985) Effect of Zn-DTPA therapy on the maternal transfer of 241Am or 237Pu to young mice. Health Phys 49:405-10

Lloyd, R D; Mays, C W; Jones, C W et al. (1985) Effect of age on the efficacy of Zn-diethylenetriaminepentaacetic acid therapy for removal of Am and Pu from beagles. Radiat Res 101:451-9